P-Dioxanone Explained

p-Dioxanone (1,4-dioxan-2-one) is the lactone of 2-(2-hydroxyethoxy)acetic acid. It is a monomer that can undergo ring-opening polymerization to give polydioxanone, a biodegradable implant material.[1] It is isomeric to trimethylene carbonate (1,3-dioxan-2-one).

Preparation

The common synthetic process for p-dioxanone is continuous gas-phase dehydrogenation of diethylene glycol on a copper or copper chromite catalyst at 280 °C.

This gives yields of up to 86%. Removal of excess diethylene glycol is crucial to the stability of the product as a monomer.[2] Further purification with recrystallization, vacuum distillation,[3] or melt crystallization allows purities of >99.5% to be achieved.

Properties

Pure p-dioxanone is a white crystalline solid with a melting point of 28 °C.[4]

Uses

The oxidation of p-dioxanone with nitric acid or dinitrogen tetroxide gives diglycolic acid at 75% yield.[5]

p-Dioxanone can undergo ring-opening polymerization catalyzed by organic compounds of tin, such as tin(II) octoate[6] or dibutyltin dilaurate, or by basic alkoxides such as aluminium isopropoxide. This affords polydioxanone, a biodegradable, semicrystalline and thermally labile polymer with uses in industry and medicine.[7] Depolymerization back to the monomer is triggered at 100 °C.

Notes and References

  1. Book: Polymeric Biomaterials in Tissue Engineering and Regenerative Medicine . Natural and Synthetic Biomedical Polymers . 20 February 2014 . Elsevier Science . 978-0-12-396983-5 . Sangamesh Kumbar, Cato Laurencin and Meng Deng.
  2. US. 5675022. Recovery of dioxanone by melt crystallization. 1995-08-23. 1997-10-07.
  3. US. 2142033. Process for the production of 2-p-dioxanone. 1936-07-01. 1938-10-27.
  4. Lee . Sang-Won . Kim . Sung-Il . Park . So-Jin . 2008 . Solubility and density of p-dioxanone in organic solvent systems . J. Korean Oil Chem. Soc. . 25 . 4 . 429–437.
  5. US. 3952054. Process for preparing diglycolic acid. 1976-04-20. Shen. C.Y..
  6. US. 3645941. Method of preparing 2-p-dioxanone polymers. 1972-02-09.
  7. Book: Bezwada . R.S. . Handbook of biodegradable polymers . Jamiolkowski . D.D. . Cooper . K. . 1997 . Harwood Academic Publishers . A. J. Domb, Joseph Kost, David M. Wiseman . 90-5702-153-6 . Australia . 29–61 . Poly(p-dioxane) and its copolymers . 38861271.