Cyclobutadieneiron tricarbonyl explained

Cyclobutadieneiron tricarbonyl is an organoiron compound with the formula Fe(C4H4)(CO)3. It is a yellow oil that is soluble in organic solvents. It has been used in organic chemistry as a precursor for cyclobutadiene, which is an elusive species in the free state.[1]

Preparation and structure

Cyclobutadieneiron tricarbonyl was first prepared in 1965 by Pettit from 3,4-dichlorocyclobutene and diiron nonacarbonyl:[2] [3]

C4H4Cl2 + 2 Fe2(CO)9 → (C4H4)Fe(CO)3 + 2 Fe(CO)5 + 5 CO + FeCl2The compound is an example of a piano stool complex. The C-C distances are 1.426 Å.[4]

Properties

Oxidative decomplexation of cyclobutadiene is achieved by treating the tricarbonyl complex with ceric ammonium nitrate. The released cyclobutadiene is trapped with a quinone, which functions as a dienophile.[5]

Cyclobutadieneiron tricarbonyl displays aromaticity as evidenced by some of its reactions, which can be classified as electrophilic aromatic substitution:[6]

It undergoes Friedel-Crafts acylation with acetyl chloride and aluminium chloride to give the acyl derivative 2, with formaldehyde and hydrochloric acid to the chloromethyl derivative 3, in a Vilsmeier-Haack reaction with N-methylformanilide and phosphorus oxychloride to the formyl 4, and in a Mannich reaction to amine derivative 5.

The reaction mechanism is identical to that of EAS:

Related compounds

Several years before Petit's work, (C4Ph4)Fe(CO)3 had been prepared from the reaction of iron carbonyl and diphenylacetylene.[7]

(Butadiene)iron tricarbonyl is isoelectronic with cyclobutadieneiron tricarbonyl.

History

In 1956, Longuet-Higgins and Orgel[8] predicted the existence of transition-metal cyclobutadiene complexes, in which the degenerate eg orbital of cyclobutadiene has the correct symmetry for π interaction with the dxz and dyz orbitals of the proper metal. The compound was synthesized three years after the prediction[9] This is a case of theory before experiment.[10]

Notes and References

  1. 10.1021/om020946c . (Cyclobutadiene)iron Tricarbonyl. A Case of Theory before Experiment . 2003 . Seyferth . Dietmar . Organometallics . 22 . 2–20 .
  2. Cyclobutadiene- and Benzocyclobutadiene-Iron Tricarbonyl Complexes G. F. Emerson, L. Watts, R. Pettit; J. Am. Chem. Soc.; 1965; 87(1); 131-133. First Page
  3. R.. Pettit. J.. Henery. 10.15227/orgsyn.050.0021. Cyclobutadieneiron Tricarbonyl. Organic Syntheses. 1970. 50. 21.
  4. . 27 . 1 . 1988 . 57–59 . 10.1021/ic00274a013 . Structure of tricarbonyl(η4-cyclobutadienyl)iron(0) at −45 °C . P. D. Harvey . W. P. Schaefer . H. B. Gray . D. F. R. Gilson . I. S. Butler.
  5. Cyclobutadiene In Synthesis: endo-Tricyclo[4.4.0.02,5]deca-3,8-diene-7,10-dione . L. Brener . J. S. Mckennis . R. Pettit. Org. Synth.. 1976. 55. 43. 10.15227/orgsyn.055.0043.
  6. Cyclobutadieneiron Tricarbonyl. A New Aromatic System J. D. Fitzpatrick, L. Watts, G. F. Emerson, R. Pettit J. Am. Chem. Soc.; 1965, vol. 87, 3254-3255 Abstract
  7. R. P. Dodge, V. Schomaker, "Crystal Structure of Tetraphenylcyclobutadiene Iron Tricarbonyl", Nature 1960, vol. 186, 798-799.
  8. Longuet-Higgins . H. C. . Orgel . L. E. . 1956-01-01 . 385. The possible existence of transition-metal complexes of cyclobutadiene . Journal of the Chemical Society (Resumed) . en . 1969–1972 . 10.1039/JR9560001969 . 0368-1769.
  9. Criegee . R. . Schröder . G. . 1959-01-21 . Ein Nickel-Komplex des Tetramethyl-Cyclobutadiens . Angewandte Chemie . de . 71 . 2 . 70–71 . 10.1002/ange.19590710210.
  10. Seyferth . Dietmar . 2003-01-01 . (Cyclobutadiene)iron TricarbonylA Case of Theory before Experiment . Organometallics . en . 22 . 1 . 2–20 . 10.1021/om020946c . 0276-7333.