SDB-005 explained

SDB-005 is an indazole-based synthetic cannabinoid that has been sold online as a designer drug.[1] It is presumed to be an agonist of the CB1 and CB2 cannabinoid receptors. SDB-005 is the indazole core analog of PB-22 where the 8-hydroxyquinoline has also been replaced with a naphthalene group.

The code number SDB-005 was originally used for a different compound, the N-phenyl instead of N-benzyl analogue of SDB-006. This compound is a potent agonist of the CB1 receptor (Ki = 21 nM) and CB2 receptor (Ki = 140 nM).[2]

However, SDB-005 was subsequently used as the name for the indazole-3-carboxylate compound mentioned above when it was sold in Europe as a designer drug, and was entered into the EMCDDA synthetic drug database under this name.[3] Consequently, there are now two distinct, yet fairly closely related cannabinoid compounds, which may both be referred to under the code SDB-005.

See also

Notes and References

  1. Web site: SDB-005 . Cayman Chemical . 27 June 2015.
  2. Banister SD, Wilkinson SM, Longworth M, Stuart J, Apetz N, English K, Brooker L, Goebel C, Hibbs DE, Glass M, Connor M, McGregor IS, Kassiou M . 6 . The synthesis and pharmacological evaluation of adamantane-derived indoles: cannabimimetic drugs of abuse . ACS Chemical Neuroscience . 4 . 7 . 1081–92 . July 2013 . 23551277 . 3715837 . 10.1021/cn400035r .
  3. https://forum.goeg.at/EwsForum/default.aspx?g=posts&t=205 EWS_EU: Neue Psychoaktive Substanzen, April 2015