Mequinol Explained

Mequinol, MeHQ or 4-methoxyphenol, is an organic compound with the formula . It is a phenol with a methoxy group in the para position. A colorless solid, it is used in dermatology[1] and organic chemistry.

Use in dermatology

Mequinol is a common active ingredient in topical drugs used for skin depigmentation. As a topical drug mequinol is often mixed with tretinoin, a topical retinoid. A common formulation for this drug is an ethanolic solution of 2% mequinol and 0.01% tretinoin by mass. Dermatologists commonly prescribe the drug to treat liver spots.

Lower dosages of mequinol have been used in conjunction with a Q-switched laser to depigment skin in patients with disseminated idiopathic vitiligo.[2]

Organic chemistry

In organic chemistry 4-methoxyphenol is used as a polymerisation inhibitor (e.g. acrylates or styrene monomers).

4-Methoxyphenol can be produced from p-benzoquinone and methanol via a free radical reaction.[3] [4]

Safety

The U.S. National Institute for Occupational Safety and Health (NIOSH) has set a recommended exposure limit (REL) of 5 mg/m3 over an 8-hour workday.[5]

See also

External links

Notes and References

  1. Web site: Stiefel Laboratories, Inc. . Full Prescribing Information . US Food and Drug Administration . 2 January 2015 .
  2. Komen L, Zwertbroek L, Burger SJ, van der Veen JP, de Rie MA, Wolkerstorfer A . Q-switched laser depigmentation in vitiligo, most effective in active disease . The British Journal of Dermatology . 169 . 6 . 1246–51 . December 2013 . 23909405 . 10.1111/bjd.12571 . 43542975 .
  3. Gambarotti C, Melone L, Punta C, Shisodia SU . Selective Monoetherification of 1,4-Hydroquinone Promoted by NaNO2 . Current Organic Chemistry . 2013 . 17 . 10 . 1108–1113 . 10.2174/1385272811317100011.
  4. Correale M, Panseri P, Romano U, Minisci F . Process for the preparation of mono-ethers of hydroquinones . US . 4933504.
  5. Web site: CDC . NIOSH Pocket Guide to Chemical Hazards . 4-Methoxyphenol . 2015-11-20 .