Isoglutamine Explained

Isoglutamine or α-glutamine is a gamma amino acid derived from glutamic acid by substituting the carboxyl group in position 1 with an amide group.[1] This is in contrast to the proteinogenic amino acid glutamine, which is the 5-amide of glutamic acid.

Isoglutamine can form the C-terminus of a peptide chain, as in muramyl dipeptide (MDP), a constituent of bacterial cell walls. It can also occur inside a peptide chain, in which case the chain is continued at the carboxyl group and isoglutamine behaves as a γ-amino acid, as in mifamurtide, a synthetic derivative of MDP used to treat osteosarcoma.

Stereochemistry

Substituting -glutamic acid, the proteinogenic enantiomer, gives -isoglutamine, which has S configuration. -Isoglutamine, the derivative of the nonproteinogenic -glutamic acid, has R configuration.[2] The latter is the form occurring in MDP and mifamurtide.

Notes and References

  1. Web site: Drugs.com: Isoglutamine . 2018-01-23 . 2018-09-20 . https://web.archive.org/web/20180920172543/https://www.drugs.com/dict/isoglutamine.html . dead .
  2. Brundish. D. E.. Wade. R.. Synthesis of N-[2-<sup>3</sup>H]acetyl-D-muramyl-L-alanyl-D-iso-glutaminyl-L-alanyl-2-(1',2'-dipalmitoyl-sn-glycero-3'-phosphoryl)ethylamide of high specific radioactivity. J Label Compd Radiopharm. 22. 1. 1985. 29–35. 10.1002/jlcr.2580220105.