Isodiazomethane Explained

In organic chemistry, isodiazomethane, also known as isocyanamide, aminoisonitrile, or systematically as isocyanoamine,[1] is the parent compound of a class of derivatives of general formula R2N–NC. It has the condensed formula H2N–N+≡C, making it an isomer of diazomethane. It is prepared by protonating an ethereal solution of lithiodiazomethane, LiCHN2, with aqueous NaH2PO4 or NH4Cl.[2] The parent compound is only marginally stable at room temperature and is isolated by removal of solvent at –50 °C.[3] Derivatives are generally prepared by dehydration of the corresponding substituted formylhydrazine with COCl2 and Et3N.[4]

Earlier, the compound was misidentified as the isomeric nitrilimine, HN–N+≡CH. However, this structure was disproven by 1H NMR studies, which show a compound with a single signal at δ 6.40 ppm in (CD3CD2)2O instead of two signals expected for nitrilimine. Moreover, an infrared band at 2140 cm−1 was assigned to the isocyano group. Transition metal complexes of isodiazomethane have been prepared.[5] In bulk form isodiazomethane is a liquid which decomposes when the temperature exceeds 15 °C. If it is heated to 40 °C, the substance explodes.[6] A solution of isodiazomethane in diethyl ether at –30 °C gradually isomerizes to diazomethane upon exposure to sodium hydroxide for 20 min.

Microwave spectroscopy indicates that unlike diazomethane, isodiazomethane is not completely planar, with the amino nitrogen undergoing inversion.[7] An ab initio study indicated that there is some N–N double bond character in H2N–N≡C, although less so than in the N–C bond of H2N–C≡N.[8] Like other isocyanide derivatives and carbon monoxide, its primary resonance form carries a negative charge and lone pair on carbon, a comparatively rare situation for neutral molecules. A resonance form with zero formal charge on all atoms also has some importance; however, the carbon atom only has a sextet of electrons and is formally a carbene.

Notes and References

  1. Web site: Aminoazaniumylidynemethane. Pubchem. pubchem.ncbi.nlm.nih.gov. en. 2018-12-21.
  2. 2012-07-29. N-Isocyanides—synthesis and reactions. Tetrahedron. en. 68. 30. 5949–5967. 10.1016/j.tet.2012.04.099. 0040-4020. Moderhack. Dietrich.
  3. Anselme. J. P.. 1966-11-01. The chemistry of isodiazomethane. Journal of Chemical Education. 43. 11. 596. 10.1021/ed043p596. 1966JChEd..43..596A. 0021-9584.
  4. Anselme. J.-P.. 1977-05-01. Isodiazomethane revisited. N-aminoisonitriles. Journal of Chemical Education. 54. 5. 296. 10.1021/ed054p296. 1977JChEd..54..296A. 0021-9584.
  5. Fehlhammer. Wolf Peter. Buračas. Peter. Bartel. Klaus. 1977. Isodiazomethane Complexes. Angewandte Chemie International Edition in English. 16. 10. 707. 10.1002/anie.197707071. 1521-3773.
  6. Book: Bretherick . L. . Bretherick's Handbook of Reactive Chemical Hazards . 2013 . Butterworth-Heinemann . 9781483284668 . 147 . en.
  7. Schäfer. Eckhard. Winnewisser. Manfred. Christiansen. Jørn Johs.. 15 July 1981. Millimeter-wave spectrum of isocyanamide, H2N-NC. Chemical Physics Letters. 81. 2. 380–386. 10.1016/0009-2614(81)80273-4. 1981CPL....81..380S.
  8. Ichikawa. Kazuo. Hamada. Yoshiaki. Sugawara. Yoko. Tsuboi. Masamichi. 15 November 1982. Ab initio study on cyanamide and isocyanamide. Chemical Physics. 72. 3. 301–312. 10.1016/0301-0104(82)85127-6. 1982CP.....72..301I.