Desulfonation reaction explained

See also: Aromatic sulfonation.

In organic chemistry, the desulfonation reaction is the hydrolysis of sulfonic acids:

RC6H4SO3H + H2O → RC6H5 + H2SO4

The reaction applied to aryl and naphthylsulfonic acids. It is the reverse of sulfonation.[1] The temperature of desulfonation correlates with the ease of the sulfonation.

Applications in synthesis

This reactivity is exploited in the regiospecific preparation of many di- and tri-substituted aromatic compounds. The approach exploits the meta-directing effect of the sulfonic acid group. 2-Chlorotoluene for example can be prepared by chlorination of p-toluenesulfonic acid, followed by hydrolysis. The method is also useful for the preparation of 2,6-dinitroaniline[2] and 2-bromophenol via phenol-2,4-disulfonic acid.[3]

References

  1. Otto Lindner, Lars Rodefeld "Benzenesulfonic Acids and Their Derivatives" in Ullmann's Encyclopedia of Industrial Chemistry 2005, Wiley-VCH, Weinheim.
  2. 2,6-Dintroaniline. Harry P. Schultz. Org. Synth.. 1951. 31. 45. 10.15227/orgsyn.031.0045.
  3. o-Bromophenol. Ralph C. Huston . Murel M. Ballard. Org. Synth.. 1934. 14. 14. 10.15227/orgsyn.014.0014.