CP 55,244 explained

CP 55,244 is a chemical compound which is a cannabinoid receptor agonist. It has analgesic effects and is used in scientific research. It is an extremely potent CB1 full agonist with a Ki of 0.21 nM, making it more potent than the commonly used full agonist HU-210.[1] [2]

See also

Notes and References

  1. Melvin LS, Milne GM, Johnson MR, Wilken GH, Howlett AC . Structure-activity relationships defining the ACD-tricyclic cannabinoids: cannabinoid receptor binding and analgesic activity . Drug Design and Discovery . 13 . 2 . 155–66 . November 1995 . 8872458 .
  2. Griffin G, Wray EJ, Martin BR, Abood ME . Cannabinoid agonists and antagonists discriminated by receptor binding in rat cerebellum . British Journal of Pharmacology . 128 . 3 . 684–8 . October 1999 . 10516649 . 1571656 . 10.1038/sj.bjp.0702806 .

This article is licensed under the GNU Free Documentation License. It uses material from the Wikipedia article "CP 55,244".

Except where otherwise indicated, Everything.Explained.Today is © Copyright 2009-2024, A B Cryer, All Rights Reserved. Cookie policy.