CP-1414S explained

CP-1414S is an experimental drug first made by a team in Germany.[1] It is a benzodiazepine derivative. CP-1414S is a 1,5-benzodiazepine, with the nitrogen atoms located at positions 1 and 5 of the diazepine ring, and so is most closely related to other 1,5-benzodiazepines such as clobazam.

CP-1414S has primarily anxiolytic and anticonvulsant effects.[2] Its potency is roughly equal to that of clobazam, but with more pronounced sedation.[3]

See also

Notes and References

  1. US Patent 3766169 PROCESS FOR THE PREPARATION OF 3-AMINOMETHYLIDENE-1,5-BENZODIAZEPINE-2,4-(3H,5H)-DIONES
  2. Carli M, Ballabio M, Caccia S, Garattini S, Samanin R . Studies on some pharmacological activities of 7-nitro-2-amino-5-phenyl-3H-1,5-benzodiazepine (CP 1414 S) in the rat. A comparison with diazepam . Arzneimittel-Forschung . 31 . 10 . 1721–3 . 1981 . 6119091 .
  3. Mennini T, Garattini S . Benzodiazepine receptors': correlation with pharmacological responses in living animals . Life Sciences . 31 . 19 . 2025–35 . November 1982 . 6129557 . 10.1016/0024-3205(82)90094-7.

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