Amfecloral Explained

Amfecloral (INN), also known as amphecloral (USAN), is a stimulant drug of the phenethylamine and amphetamine chemical classes that was used as an appetite suppressant under the trade name Acutran, but is now no longer marketed.[1] It was classified as an anorectic drug with little to no stimulant activity in a 1970 review.[2] The British Pharmacopoeia Commission approved the name in 1970.[3] The raw ingredients used in manufacturing it were d-amphetamine and chloral hydrate.[4]

Pharmacology

Amfecloral is metabolised to both d-(S)- and l-(R)-amphetamine and, most likely, also to chloral hydrate.[5] Amphetamine is a psychostimulant, whereas chloral hydrate is a sedative/hypnotic drug.

The extent of metabolism and in-vivo contribution of a chloral hydrate metabolism to its purported "little to no stimulant activity" is unknown.

See also

Notes and References

  1. Book: Dictionary of pharmacological agents, Volumes 1-2 . Ganellin CR, Triggle DJ . 1996 . Chapman & Hall . 9780412466304 . 67 .
  2. Van Rossum JM . Mode of action of psychomotor stimulant drugs . International Review of Neurobiology . 12 . 307–83 . 1970 . 4918147 . 10.1016/s0074-7742(08)60065-3 . 9780123668127 .
  3. Notes and News. The Lancet. October 1970. 296. 7675. 730–732. 10.1016/S0140-6736(70)92010-6.
  4. Book: McPherson. Edwin M. . vanc . Pharmaceutical Manufacturing Encyclopedia . 2007 . Elsevier . Burlington . 9780815518563 . 244 . 3rd .
  5. Web site: NCATS Inxight Drugs — AMFECLORAL, (+)- . 2024-07-16 . drugs.ncats.io . en.